Linagliptin

Name: Linagliptin
Brand: Vaqora Chemicals
SKU: VQ-007545

About Linagliptin

Listed under CAS 668270-12-0, Linagliptin is a high-purity reference standard of Linagliptin available from Vaqora Chemicals. With the molecular formula C25H28N8O2, it has a molar mass of 472.5 g/mol. Its systematic (IUPAC) name is 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione. It is also known as BI 1356BS or BI-1356-BS.

The product is provided as a solid. Reference materials should be stored sealed and away from light and moisture, as specified on the accompanying COA. Handle it with standard laboratory precautions and appropriate personal protective equipment.

Laboratories use this Linagliptin standard for identity and assay testing, system suitability checks and method validation supporting ANDA and DMF filings. Typical end-use sectors are pharmaceutical manufacturing and academic and industrial research.

Vaqora Chemicals supplies Linagliptin in 10 mg, 25 mg, 50 mg and 100 mg packs, each shipped with a Certificate of Analysis (COA), and exports worldwide. This item is currently in stock for prompt dispatch.

Typical applications

Identification & assay
Method development & validation
QC reference material

Industries

Related to Linagliptin

View every impurity, metabolite and intermediate we list for Linagliptin.

Linagliptin impurities

Specifications & identifiers

Chemical identifiers
Product name	Linagliptin
Catalogue No.	VQ-007545
CAS Number	668270-12-0
Other CAS	1233245-20-9, 1233245-11-8
IUPAC name	8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione
Molecular formula	C₂₅H₂₈N₈O₂
Molecular weight	472.5 g/mol
Exact mass	472.2335
Grade	Reference Standard
HSN code	38229090
InChIKey	LTXREWYXXSTFRX-QGZVFWFLSA-N
SMILES	CC#CCN1C2=C(N=C1N3CCC[C@H](C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C
PubChem CID	10096344

Physical properties
Physical form	Solid
LogP (XLogP3)	1.9
H-bond donors / acceptors	1 / 7
TPSA	113 Å²
Synonyms	BI 1356BS, BI-1356-BS, linagliptine, BS 1356 BS, BI-1356BS, BI 1356 BS, BS-1356-BS, 1356, BI, Linagliptin (BI-1356), ione, Linaglitpin, Tradjenta (TN)

Documents

Safety Data Sheet (SDS)16-section GHS · on request Certificate of AnalysisTypical / batch COA · on request Specification sheetTDS / MOA · on request

Frequently asked questions

What is the CAS number of Linagliptin?

The CAS Registry Number of Linagliptin is 668270-12-0. It is also known as BI 1356BS, BI-1356-BS, linagliptine.

What is the molecular formula and molecular weight of Linagliptin?

Linagliptin has the molecular formula C25H28N8O2 and a molecular weight of 472.5 g/mol. Its IUPAC name is 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione.

What is Linagliptin used for?

Linagliptin is supplied as a characterised reference material related to Linagliptin. It is used for analytical method development and validation (AMV), impurity profiling, stability studies and quality control, and in ANDA/DMF regulatory filings.

Which grade and pack sizes of Linagliptin can I order?

We supply Linagliptin in Reference Standard grade, in 10 mg, 25 mg, 50 mg, 100 mg packs. Larger bulk quantities and custom packing are quoted on request.

Do you provide a COA and SDS with Linagliptin?

Yes. Every lot of Linagliptin is shipped with a batch-specific Certificate of Analysis, and a 16-section GHS Safety Data Sheet is provided with the quotation and the shipment.

Can Linagliptin be shipped internationally?

Yes. We export Linagliptin worldwide by air and sea freight or express courier, on EXW, FOB, CIF, CFR or DAP Incoterms, with full export documentation.