Pelitinib

Name: Pelitinib
Brand: Vaqora Chemicals
SKU: VQ-043763

About Pelitinib

Listed under CAS 257933-82-7, Pelitinib is a high-purity reference standard of Pelitinib available from Vaqora Chemicals. With the molecular formula C24H23ClFN5O2, it has a molar mass of 467.9 g/mol. Its systematic (IUPAC) name is (E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide. It is also known as EKB-569 or EKB 569.

The product is provided as a solid. Keep the vial tightly closed, protected from light and humidity, at the temperature stated on the Certificate of Analysis. Under GHS it is labelled “Danger”, so handle it with suitable PPE and consult the SDS.

As a reference sample of Pelitinib, it is used for identification, assay and impurity-profiling work during analytical method development, validation (AMV) and routine QC. Our customers for this product work in pharmaceutical manufacturing and academic and industrial research.

Standard pack sizes are 10 mg, 25 mg, 50 mg and 100 mg, and every batch ships with a Certificate of Analysis (COA) and we export worldwide.

Typical applications

Identification & assay
Method development & validation
QC reference material

Industries

Related to Pelitinib

View every impurity, metabolite and intermediate we list for Pelitinib.

Pelitinib impurities

Specifications & identifiers

Chemical identifiers
Product name	Pelitinib
Catalogue No.	VQ-043763
CAS Number	257933-82-7
IUPAC name	(E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide
Molecular formula	C₂₄H₂₃ClFN₅O₂
Molecular weight	467.9 g/mol
Exact mass	467.1524
Grade	Reference Standard
HSN code	38229090
InChIKey	WVUNYSQLFKLYNI-AATRIKPKSA-N
SMILES	CCOC1=C(C=C2C(=C1)N=CC(=C2NC3=CC(=C(C=C3)F)Cl)C#N)NC(=O)/C=C/CN(C)C
PubChem CID	6445562

Physical properties
Physical form	Solid
LogP (XLogP3)	4.5
H-bond donors / acceptors	2 / 7
TPSA	90.3 Å²
Synonyms	EKB-569, EKB 569, EKI 569, Pelitinib (EKB-569), EKI-569, 2-Butenamide, (E)-,, 4-chloro-2-amino-benzoic ac, EX-A061

Safety & hazard information (GHS)

Toxic

Signal word: Danger

Hazard statements

H301Toxic if swallowed

Precautionary statements: P264, P270, P301 + P316, P321, P330, P405, P501

Classification is indicative (aggregated GHS notifications) and may vary by grade and concentration. Always refer to the SDS supplied with your lot.

Documents

Safety Data Sheet (SDS)16-section GHS · on request Certificate of AnalysisTypical / batch COA · on request Specification sheetTDS / MOA · on request

Frequently asked questions

What is the CAS number of Pelitinib?

The CAS Registry Number of Pelitinib is 257933-82-7. It is also known as EKB-569, EKB 569, EKI 569.

What is the molecular formula and molecular weight of Pelitinib?

Pelitinib has the molecular formula C24H23ClFN5O2 and a molecular weight of 467.9 g/mol. Its IUPAC name is (E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide.

What is Pelitinib used for?

Pelitinib is supplied as a characterised reference material related to Pelitinib. It is used for analytical method development and validation (AMV), impurity profiling, stability studies and quality control, and in ANDA/DMF regulatory filings.

Which grade and pack sizes of Pelitinib can I order?

We supply Pelitinib in Reference Standard grade, in 10 mg, 25 mg, 50 mg, 100 mg packs. Larger bulk quantities and custom packing are quoted on request.

Do you provide a COA and SDS with Pelitinib?

Yes. Every lot of Pelitinib is shipped with a batch-specific Certificate of Analysis, and a 16-section GHS Safety Data Sheet is provided with the quotation and the shipment.

Can Pelitinib be shipped internationally?

Yes. Pelitinib is classified as hazardous, so it is packed in UN-approved packaging and shipped as dangerous goods under IATA/IMDG rules. We export worldwide on EXW, FOB, CIF and DAP terms.