Gilteritinib

Name: Gilteritinib
Brand: Vaqora Chemicals
SKU: VQ-007494

About Gilteritinib

Listed under CAS 1254053-43-4, Gilteritinib is a high-purity reference standard of Gilteritinib available from Vaqora Chemicals. Formula C29H44N8O3, molecular weight 552.7 g/mol. Common synonyms include ASP-2215 and ASP 2215.

The product is provided as a solid. Reference materials should be stored sealed and away from light and moisture, as specified on the accompanying COA. The GHS classification uses the signal word “Danger”, so appropriate gloves, eye protection and ventilation are recommended.

Laboratories use this Gilteritinib standard for identity and assay testing, system suitability checks and method validation supporting ANDA and DMF filings. Typical end-use sectors are pharmaceutical manufacturing and academic and industrial research.

Available in 10 mg, 25 mg, 50 mg and 100 mg packs, Gilteritinib is dispatched with a Certificate of Analysis (COA) to destinations worldwide. Stock is available for quick dispatch.

Typical applications

Identification & assay
Method development & validation
QC reference material

Industries

Related to Gilteritinib

View every impurity, metabolite and intermediate we list for Gilteritinib.

Gilteritinib impurities

Specifications & identifiers

Chemical identifiers
Product name	Gilteritinib
Catalogue No.	VQ-007494
CAS Number	1254053-43-4
IUPAC name	6-ethyl-3-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide
Molecular formula	C₂₉H₄₄N₈O₃
Molecular weight	552.7 g/mol
Exact mass	552.3536
Grade	Reference Standard
HSN code	38229090
InChIKey	GYQYAJJFPNQOOW-UHFFFAOYSA-N
SMILES	CCC1=C(N=C(C(=N1)C(=O)N)NC2=CC(=C(C=C2)N3CCC(CC3)N4CCN(CC4)C)OC)NC5CCOCC5
PubChem CID	49803313

Physical properties
Physical form	Solid
LogP (XLogP3)	3.5
H-bond donors / acceptors	3 / 10
TPSA	121 Å²
Synonyms	ASP-2215, ASP 2215, Gilteritinib HCl, C6F, Gilteritinib (Standard), Gilteritinib(ASP2215), Gilteritinib (USAN/INN), ASP2215 (Gilteritinib), Gilteritinib(ASP2215)?, Gilteritinib (ASP-2215), EX-A2775

Safety & hazard information (GHS)

Health hazard

Signal word: Danger

Hazard statements

H360May damage fertility or the unborn child
H373May causes damage to organs through prolonged or repeated exposure

Precautionary statements: P203, P260, P280, P318, P319, P405, P501

Classification is indicative (aggregated GHS notifications) and may vary by grade and concentration. Always refer to the SDS supplied with your lot.

Documents

Safety Data Sheet (SDS)16-section GHS · on request Certificate of AnalysisTypical / batch COA · on request Specification sheetTDS / MOA · on request

Frequently asked questions

What is the CAS number of Gilteritinib?

The CAS Registry Number of Gilteritinib is 1254053-43-4. It is also known as ASP-2215, ASP 2215, Gilteritinib HCl.

What is the molecular formula and molecular weight of Gilteritinib?

Gilteritinib has the molecular formula C29H44N8O3 and a molecular weight of 552.7 g/mol. Its IUPAC name is 6-ethyl-3-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide.

What is Gilteritinib used for?

Gilteritinib is supplied as a characterised reference material related to Gilteritinib. It is used for analytical method development and validation (AMV), impurity profiling, stability studies and quality control, and in ANDA/DMF regulatory filings.

Which grade and pack sizes of Gilteritinib can I order?

We supply Gilteritinib in Reference Standard grade, in 10 mg, 25 mg, 50 mg, 100 mg packs. Larger bulk quantities and custom packing are quoted on request.

Do you provide a COA and SDS with Gilteritinib?

Yes. Every lot of Gilteritinib is shipped with a batch-specific Certificate of Analysis, and a 16-section GHS Safety Data Sheet is provided with the quotation and the shipment.

Can Gilteritinib be shipped internationally?

Yes. Gilteritinib is classified as hazardous, so it is packed in UN-approved packaging and shipped as dangerous goods under IATA/IMDG rules. We export worldwide on EXW, FOB, CIF and DAP terms.