Saxagliptin

Name: Saxagliptin
Brand: Vaqora Chemicals
SKU: VQ-004144

About Saxagliptin

Vaqora Chemicals supplies Saxagliptin in IP/BP/USP grade, a metabolic / hormonal API registered under CAS number 361442-04-8. Its molecular formula is C18H25N3O2 and its molecular weight is 315.4 g/mol. Systematically, it is named (1S,3S,5S)-2-[(2S)-2-amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile. It is also known as Saxagliptin anhydrous or Saxagliptine.

It is supplied as a powder. Store sealed in a dry, well-ventilated location away from incompatible materials. The GHS classification uses the signal word “Danger”, so appropriate gloves, eye protection and ventilation are recommended.

This API belongs to our antidiabetic, hormone and metabolic APIs portfolio and is supplied to IP/BP/USP specifications for formulators, contract manufacturers and generic drug developers. Typical end-use sectors are pharmaceutical manufacturing.

Standard pack sizes are 1 kg, 5 kg and 25 kg, and every batch ships with a Certificate of Analysis (COA) and we export worldwide.

Typical applications

Pharmaceutical synthesis
Pharmaceutical formulation

Industries

Related to Saxagliptin

View every impurity, metabolite and intermediate we list for Saxagliptin.

Saxagliptin impurities

Grade guides

Specifications & identifiers

Chemical identifiers
Product name	Saxagliptin
Catalogue No.	VQ-004144
CAS Number	361442-04-8
IUPAC name	(1S,3S,5S)-2-[(2S)-2-amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile
Molecular formula	C₁₈H₂₅N₃O₂
Molecular weight	315.4 g/mol
Exact mass	315.1947
Grade	IP/BP/USP
HSN code	2933
InChIKey	QGJUIPDUBHWZPV-SGTAVMJGSA-N
SMILES	C1[C@@H]2C[C@@H]2N([C@@H]1C#N)C(=O)[C@H](C34CC5CC(C3)CC(C5)(C4)O)N
PubChem CID	11243969

Physical properties
Physical form	Powder
LogP (XLogP3)	0.7
H-bond donors / acceptors	2 / 4
TPSA	90.4 Å²
Synonyms	Saxagliptin anhydrous, Saxagliptine, 3-hydroxyadamantylglycine-4,5-methanoprolinenitrile hydrate, Saxagliptin Monohydrate, OPC-262, OPC 262, Saxagliptin (USAN/INN), Saxagliptin for system suitability CRS, (S)-3-Hydroxyadamantylglycine-L-cis-4,5-methanoprolinenitrile TFA salt, (1S,6S)-2-(2-adamantan-1-yl-2-amino-acetyl)-2-aza-bicyclo[3.1.0]hexane-3-carbonitrile

Safety & hazard information (GHS)

Health hazard

Signal word: Danger

Hazard statements

H317May cause an allergic skin reaction
H334May cause allergy or asthma symptoms or breathing difficulties if inhaled
H372Causes damage to organs through prolonged or repeated exposure

Precautionary statements: P203, P233, P260, P261, P264, P270, P271, P272, P280, P284, P302 + P352, P304 + P340, P318, P319, P321, P333 + P317, P342 + P316, P362 + P364, P403, P405, P501

Classification is indicative (aggregated GHS notifications) and may vary by grade and concentration. Always refer to the SDS supplied with your lot.

Documents

Safety Data Sheet (SDS)16-section GHS · on request Certificate of AnalysisTypical / batch COA · on request Specification sheetTDS / MOA · on request

Other grades of CAS 361442-04-8

Reference Standard

Saxagliptin WS

CAS: 361442-04-8
Formula: C₁₈H₂₅N₃O₂
MW: 315.4 g/mol

In stock

Frequently asked questions

What is the CAS number of Saxagliptin?

The CAS Registry Number of Saxagliptin is 361442-04-8. It is also known as Saxagliptin anhydrous, Saxagliptine, 3-hydroxyadamantylglycine-4,5-methanoprolinenitrile hydrate.

What is the molecular formula and molecular weight of Saxagliptin?

Saxagliptin has the molecular formula C18H25N3O2 and a molecular weight of 315.4 g/mol. Its IUPAC name is (1S,3S,5S)-2-[(2S)-2-amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile.

What is Saxagliptin used for?

Saxagliptin is supplied as a characterised reference material related to Saxagliptin. It is used for analytical method development and validation (AMV), impurity profiling, stability studies and quality control, and in ANDA/DMF regulatory filings.

Which grade and pack sizes of Saxagliptin can I order?

We supply Saxagliptin in IP/BP/USP grade, in 1 kg, 5 kg, 25 kg packs. Larger bulk quantities and custom packing are quoted on request.

Do you provide a COA and SDS with Saxagliptin?

Yes. Every lot of Saxagliptin is shipped with a batch-specific Certificate of Analysis, and a 16-section GHS Safety Data Sheet is provided with the quotation and the shipment.

Can Saxagliptin be shipped internationally?

Yes. Saxagliptin is classified as hazardous, so it is packed in UN-approved packaging and shipped as dangerous goods under IATA/IMDG rules. We export worldwide on EXW, FOB, CIF and DAP terms.